Buy Thiamylal

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Thiamylal (Surital) is a barbiturate derivative invented in the 1950s. It has sedative, anticonvulsant, and hypnotic effects, and is used as a strong but short acting sedative. Thiamylal is still in current use, primarily for induction in surgical anaesthesia  or as an anticonvulsant to counteract side effects from other anaesthetics.It is the thiobarbiturate analogue of secobarbital.

A barbiturate that is administered intravenously for the production of complete anesthesia of short duration, for the induction of general anesthesia, or for inducing a hypnotic state.

Thiamylal, a barbiturate, is used in combination with acetaminophen or aspirin and caffeine for its sedative and relaxant effects in the treatment of tension headaches, migraines, and pain. Barbiturates act as nonselective depressants of the central nervous system (CNS), capable of producing all levels of CNS mood alteration from excitation to mild sedation, hypnosis, and deep coma. In sufficiently high therapeutic doses, barbiturates induce anesthesia.

Thiamylal binds at a distinct binding site associated with a Cl- ionopore at the GABAA receptor, increasing the duration of time for which the Cl- ionopore is open. The post-synaptic inhibitory effect of GABA in the thalamus is, therefore, prolonged.

Thiamylal sodium is a new, ultra-short-acting thiobarbiturate, which in this study was used by the intravenous route. In all cases a 2.5% solution was injected on the electroshock table immediately prior to the application of current. The administration of drug sufficient to destroy the corneal reflex was found either to eliminate the muscular contractions or so materially to reduce them that electroshock was safe, despite the presence of known fractures. The usual facial twitchings and upward movements of the eyeballs.

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